CID-1375606 is a GPR27 agonist with EC50 values of 0.46 uM and 7.9 uM in chimeric GPR27V2 and wild-type GPR27 luciferase B-arrestin-2 complementation assays, respectively.{54081} It is selective for GPR27 over the closely related receptors GPR85 and GPR173 for which it does not induce B-arrestin-2 recruitment in the same assay. GPR27 function has been linked to insulin promoter activity and excretion.{54082}
Specifications
Size
25 mg
CAS number
313493-80-0
Supplier
Cayman Chemical
Shipping & storage
Shipping condition
Dry Ice
Storage temperature
-20°C