1,2,3,4-Tetrahydrostaurosporine is a derivative of staurosporine (Item No. 81590) and an inhibitor of mutant EGFR (IC50 = 74 nM for EGFRT790M).{53434} It is selective for EGFRT790M over wild-type EGFR (IC50 = 390 nM). It also binds to Janus kinase 3 (JAK3).{53435}
Specifications
Size
1 mg
CAS number
220038-19-7
Supplier
Cayman Chemical
Shipping & storage
Shipping condition
Dry Ice
Storage temperature
-20°C